Development of one-pot benzylic amination reactions of azine N-oxides
نویسندگان
چکیده
منابع مشابه
One-pot borylation/amination reactions: syntheses of arylamine boronate esters from halogenated arenes.
[reaction: see text] A one-pot protocol for converting 1,3- and 1,4-substituted aryl halides to arylamine boronate esters is described. This is achieved by sequential Ir-catalyzed aromatic borylation at the least hindered C-H bond of the aryl halide and subsequent Pd-catalyzed C-N coupling at the halide position of the crude arylboronic ester.
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ژورنال
عنوان ژورنال: Tetrahedron Letters
سال: 2018
ISSN: 0040-4039
DOI: 10.1016/j.tetlet.2018.03.062